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- Varenicline (category 5-HT3 agonists)"Varenicline is a partial agonist at alpha4beta2 and a full agonist at alpha7 neuronal nicotinic receptors". Molecular Pharmacology. 70 (3): 801–5. doi:10.1124/mol...23 KB (2,363 words) - 18:18, 17 December 2020